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Kisspeptin-234 trifluoroacetate salt

SIGMA/K2644 - ≥95% (HPLC)

Synonym: kisspeptin-10 peptide 234

CAS Number: 1848962-29-7
Empirical Formula (Hill Notation): C63H78N18O13 · xC2HF3O2
Molecular Weight: 1295.41 (free base basis)
Linear Formula: C63H78N18O13 · xC2HF3O2
Product Type: Chemical
Catalog Number PKG Qty. Price Quantity
45-K2644-1MG 1 mg
 $184.00
1/EA		 Add To Favorites
This image is provided for informative purposes only and does not represent an actual product label. It should not be used as a substitute for official product labeling.

 

assay ≥95% (HPLC)
color colorless to white
form film
Quality Level 100 
solubility H2O: >1 mg/mL
storage temp. −20°C
Biochem/physiol Actions: Kisspeptin-234 is a 10-amino acid peptide antagonist with potent neutral antagonist activity at GPR-54 and competes directly at the Kisspeptin-10 binding site.
Biochem/physiol Actions: Kisspeptin-234 is a 10-amino acid peptide antagonist with potent neutral antagonist activity at GPR-54 and competes directly at the Kisspeptin-10 binding site. Kisspeptin-234 is the first reported antagonist for the kisspeptin-1/GPR-54 signaling system.

Gonadotropin-releasing hormone (GnRH) modulates the hypothalamic-pituitary-gonadal axis, enabling the brain to control reproductive processes. Kisspeptin-1 is a peptide neurotransmitter released from afferent neurons onto GnRH neurons, where it binds to and activates to the orphan receptor GPR-54 to regulate release of GnRH. Regulation of kisspeptin/GPR-54 signaling presents an opportunity for reproductive therapeutics above the level of GnRH and gonadotropin secretion. Pharmacological and selective tools are needed to better understand kisspeptin-1/GPR-54 signaling. Analogs of kisspeptin-10, a 10-amino acid portion of kisspeptin-1, were designed to be full and neutral antagonists of GPR-54.
Packaging: 1 mg in glass bottle
RIDADR NONH for all modes of transport
WGK Germany WGK 2
Flash Point(F) Not applicable
Flash Point(C) Not applicable
Purity ≥95% (HPLC)
Storage Temp. −20°C
UNSPSC 12352200

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